内容简介
Chapter 1 Introduction
Ⅰ.Development of Pharmacology
Ⅱ.New Drug Research
Chapter 2 Pharmacodynamics
Ⅰ.General Classification of Drug Effects
Ⅱ.Dose-Effect Relationship
Ⅲ.Receptor Theory and Drug Receptor Interaction
Ⅳ.Receptor Families and Their Transducer and Effector Molecules
Ⅴ.Relationship Between Regulatory Mechanisms of Receptors and the Pharmacological Action
Ⅵ.Mechanism of Action
Chapter 3 Pharmacokinetics
Ⅰ.Drug Transport across Membranes
Ⅱ.The Dynamics of Drug Absorption,Distribution,and Elimination
Ⅲ.General Principles of Pharmacokinetics
Chapter 4 Pharmacogenetics
Ⅰ.The Objectives of Research in Pharmacogenetics
Ⅱ.The Effect of Genetic Factors on Drug Reactions
Ⅲ.The Racial Difference of Drug Reaction and Metabolism
Chapter 5 Autonomic Pharmacology
Ⅰ.Anatomy and Neurotransmitter Chemistry of the Autonomic Nervous System
Ⅱ.Biosynthesis and Metabolism of Transmitters
Ⅲ.Locations of Autonomic Receptors
Ⅳ.Presynaptic Regulation of Transmitter Release
Ⅴ.Functional Organization of Autonomic Activity
Ⅵ.Coupling Mechanism of Receptor-effect
Ⅶ.Mode of Action of Autonomic Nervous System Drugs
Ⅷ.Classification of Autonomic Nervous System Drugs
Chapter 6 Cholinoceptor-Activating and Cholinesterase-Inhibiting Drugs
Ⅰ.Direct-acting Cholinoceptor Stimulants
Ⅱ.Cholinesterase Inhibitors
Chapter 7 Organophosphates Anticholinesterase Intoxication and Cholinesterase Reactivators
Ⅰ.Organophosphates Anticholinesterase Intoxication
Ⅱ.Cholinesterase Reactivator
Chapter 8 M Cholinoceptor Antagonists
Ⅰ.Natural M Cholinoceptor Blocking Drugs
Ⅱ.Synthetic Spasmolytic Drugs
Chapter 9 N Cholinoceptor Antagonists
Ⅰ.N1 Cholinoceptor Blocking Drugs
Ⅱ.N2 Cholinoceptor Blocking Drugs
Chapter 10 Adrenoceptor-Activating Drugs
Ⅰ.Chemical Structure
Ⅱ.Classification
Ⅲ.Mixed α and β Receptor Agonists
Ⅳ.α Receptor Agonists
Ⅴ.β Receptor Agonists
Ⅵ.Dopaminergic Receptor Agonists
Chapter 11 Adrenoceptor Blocking Drugs
Ⅰ.α Receptor Antagonists
Ⅱ.β Receptor Antagonists
Ⅲ.α,β Receptor Antagonists
Chapter 12 Sedative-Hypnotics Drugs
Ⅰ.Introduction
Ⅱ.Benzodiazepines
Ⅲ.Barbiturates
Ⅳ.Other Sedative-Hypnotics
Chapter 13 Antiepileptic Drugs
Ⅰ.Classification of Seizure Types
Ⅱ.Drugs Used in Seizures
Ⅲ.Selectivity and Withdrawal of Antiepileptic Drugs
Ⅳ.Anticonvulsant Drugs
Chapter 14 Psychotropic Drugs
Ⅰ.Antipsychotic Drugs
Ⅱ.Antimanic Drugs
Ⅲ.Antidepressants
Chapter 15 Antiparkinsonism Drugs
Ⅰ.Dopaminergic Drugs
Ⅱ.Anticholinergic Drugs
Ⅲ.Others
Chapter 16 Antipyretic-Analgesic and Antiinflammatory Drugs
Ⅰ.Introduction
Ⅱ.Salicylates
Ⅲ.Anilines
Ⅳ.Pyrazolones
Ⅴ.Others
Ⅵ.Analgesic Compounds
Ⅶ.Slow Acting Antirheumatic Drugs
Ⅷ.Antigout Drugs
Chapter 17 Narcotic Analgesics
Ⅰ.Introduction
Ⅱ.Opioid Receptor Agonists
Ⅲ.Opioid Receptor Antagonists
Chapter 18 Central Stimulants
Ⅰ.Cerebral Stimulants
Ⅱ.Medullary Stimulants
Chapter 19 Drugs Used in the Treatment of Heart Failure
Ⅰ.Pathophysiology of Congestive Heart Failure
Ⅱ.Diuretics
Ⅲ.Aldosterone Antagonists
Ⅳ.Inhibitors of RAAS:ACEI and AT1 Receptor Antagonists
Ⅴ.β Adrenergic Receptor Blocking Agents
Ⅵ.Vasodilators
Ⅶ.Cardiac Glycosides
Ⅷ.β Adrenergic Receptor Stimulators
Ⅸ.Phosphodiesterase Inhibitors
Chapter 20 Antihypertensive Drugs
Ⅰ.Introduction
Ⅱ.Drugs that Alter Sodium and Water Balance
Ⅲ.Drugs that Alter Sympathetic Nervous System Function
Ⅳ.Vasodilators
Ⅴ.Drugs that Interfere with the Renin-Angiotensin System
Ⅵ.Clinical Pharmacology of Antihypertensive Drugs
Chapter 21 Anti-Angina Pectoris Drugs
Ⅰ.Introduction
Ⅱ.Nitrates and Nitrites
Ⅲ.Calcium Channel Blockers
Ⅳ.β Receptor Antagonists
Chapter 22 Antiarhythmic Drugs
Ⅰ.Introduction
Ⅱ.Class IA
Ⅲ.Class IB
Ⅳ.Class IC
Ⅴ.Class Ⅱ
Ⅵ.Class Ⅲ
Ⅶ.Class Ⅳ
Ⅷ.Others
Chapter 23 Antihyperlipidemic Drugs
Ⅰ.Atherogenesis
Ⅱ.Lipoprotein Transport
Ⅲ.Dyslipidaemia
Ⅳ.Antihyperlipidemic Drugs
Chapter 24 Diuretic and Dehydrant Drugs
Ⅰ.Kidney Structure and Function
Ⅱ.Diuretics
Ⅲ.Osmotic Diuretics(Mannitol,Sorbitol,Glucose,Urea)
Chapter 25 Antiasthmatic Drugs
Ⅰ.Bronchodilators
Ⅱ.Anti-Inflammatory Drugs
Chapter 26 Drugs Used in Gastrointestinal Diseases
Ⅰ.Drugs Used to Treat Peptic Ulcer
Ⅱ.Antiemetic Drugs
Ⅲ.Antidiarrheal Drugs
Ⅳ.Laxatives
Chapter 27 Drugs Affecting Uterine Motility
Ⅰ.Drugs that Stimulate Uterine Contraction
Ⅱ.Drugs that Inhibit Uterine Contraction
Chapter 28 Anticoagulants and Coagulants
Ⅰ.Introduction
Ⅱ.Anticoagulants
Ⅲ.Antiplatelet Drugs
Ⅳ.Fibrinolytic Drugs
Ⅴ.Coagulants
Chapter 29 Histamine and Antihistamine Drugs
Ⅰ.Histamine
Ⅱ.H1 Receptor Antagonists
Ⅲ.H2 Receptor Antagonists
Chapter 30 Adrenocorticosteroids
Ⅰ.Introduction
Ⅱ.Glucocorticoids
Ⅲ.Mineralocorticoids
Chapter 31 Drugs Affecting the Thyroid Gland
Ⅰ.Thyroid Hormone(TH)
Ⅱ.Antithyroid Drugs
Chapter 32 Antidiabetic Drugs
Ⅰ.Insulin
Ⅱ.Oral Hypoglycemic Drugs
Ⅲ.Current Treatment Options
Chapter 33 Introduction to Antibacterial Drugs
Ⅰ.Specialty Terms
Ⅱ.Antimicrobial Mechanisms
Ⅲ.Mechanism of Resistance to Antibiotics
Chapter 34 Synthetic Antimicrobial Drugs
Ⅰ.Sulfonamides
Ⅱ.Trimethoprim
Ⅲ.Quinolones
Chapter 35 β-Lactam Antibiotics
Ⅰ.Penicillins
Ⅱ.Cephalosporins
Ⅲ.Other β-Lactam Drugs
Chapter 36 Macrolides,Lincosamides and Glycopeptides
Ⅰ.Macrolides
Ⅱ.Lincosamides
Ⅲ.Glycopeptides
Chapter 37 Broad-Spectrum Antibiotics
Ⅰ.Tetracyclines
Ⅱ.Chloramphenicols
Chapter 38 Aminoglycosides and Polypeptides
Ⅰ.Aminoglycosides
Ⅱ.Polypeptides
Chapter 39 Antifungal Drugs
Ⅰ.Antibiotics
Ⅱ.Azole Antifungal Drugs
Ⅲ.Allylamine Antifungal Drugs
Ⅳ.Pyrimidine Antifungal Drugs
Chapter 40 Antiviral Drugs
Ⅰ.Anti-Human Immunodeficiency Virus Drugs
Ⅱ.Anti-Herpersvirus Drugs
Ⅲ.Anti-Influenza Drugs
Ⅳ.Anti-Hepacivirus Drugs
Chapter 41 Antimycobacterial Drugs
Ⅰ.Introduction
Ⅱ.First-Line Drugs Used in Tuberculosis
Ⅲ.Alternative Second-Line Drugs in Treatment of Tuberculosis
Ⅳ.Combination Chemotherapy ofTuberculosis
Chapter 42 Antimalarial Drugs
Ⅰ.Plasmodium Life Cycles and Action of Antimalarial Drugs
Ⅱ.Antimalarial Drugs Mainly Applied to Control Symptoms
Ⅲ.Antimalarial Drugs Mainly Applied to Control Relapse and Transmission
Ⅳ.Antimalarial Drugs MainlyApplied to Causal Prophylaxis
Chapter 43 Amebicides
Ⅰ.Life Cycles of Entamoeba Histolytica and Action of Amebicides
Ⅱ.Luminal Amebicides
Ⅲ.Extraintestinal Amebicides
Ⅳ.Luminal and Simultaneously Extraintestinal Amebicides
Chapter 44 Anthelmintic Drugs
Ⅰ.Nematocides
Ⅱ.Taeniacides
Ⅲ.Anti-Trematode Drugs
Chapter 45 Antineoplastic Drugs
Ⅰ.Introduction
Ⅱ.Cytotoxic Drugs
Ⅲ.Non-Cytotoxic Drugs
References